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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
TGF-beta receptor type-1
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50293517
(2-(6-methylpyridin-2-yl)-N-(2-methylpyridin-4-yl)q...)
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Affinity Data
IC50: 199nM
Assay Description:
Inhibition of human ALK5 kinase expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
TGF-beta receptor type-1
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50293517
(2-(6-methylpyridin-2-yl)-N-(2-methylpyridin-4-yl)q...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.02E+3nM
Assay Description:
Inhibition of TGFbeta-induced ALK5 in human HepG2 cells by luciferase assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
TGF-beta receptor type-1
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50293517
(2-(6-methylpyridin-2-yl)-N-(2-methylpyridin-4-yl)q...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of GST-fused p38alpha
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI