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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Vasopressin V2 receptor
(Homo sapiens (Human))
Wyeth-Ayerst Research
Curated by
ChEMBL
Ligand
BDBM50065121
(CHEMBL310416 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a]...)
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Affinity Data
IC50: 1nM
Assay Description:
Displacement of [3H]-AVP from human V2 receptor expressed in murine fibroblast cell line (LV2) membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Vasopressin V2 receptor
(Rattus norvegicus (Rat))
Wyeth-Ayerst Research
Curated by
ChEMBL
Ligand
BDBM50065121
(CHEMBL310416 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a]...)
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Copy InChI
Affinity Data
IC50: 4.5nM
Assay Description:
Displacement of [3H]-AVP from vasopressin V2 receptor of rat kidney medulla.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Vasopressin V1a receptor
(RAT)
Wyeth-Ayerst Research
Curated by
ChEMBL
Ligand
BDBM50065121
(CHEMBL310416 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a]...)
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Copy InChI
Affinity Data
IC50: 54nM
Assay Description:
Displacement of (Phe-3,4,5-H) Vasopressin from V1a recptor from rat liver membranes.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Vasopressin V1a receptor
(Homo sapiens (Human))
Wyeth-Ayerst Research
Curated by
ChEMBL
Ligand
BDBM50065121
(CHEMBL310416 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a]...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 59nM
Assay Description:
Displacement of [3H]-AVP from vasopressin receptor (V1a) from human platelet membranes.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI