Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCathepsin G(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075116(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-(2-met...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against human leukocyte cathepsin G (h-CG)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen B(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075116(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-(2-met...)
Affinity DataIC50:  190nMAssay Description:Inhibitory activity against human chymase (h-chymase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-like elastase family member 2A(Sus scrofa)
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075116(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-(2-met...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory activity against porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075116(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-(2-met...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibitory activity against human chymase (h-chymase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Nippon Steel

Curated by ChEMBL
LigandPNGBDBM50075116(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-(2-met...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed