Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProstaglandin E synthase 2(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50339582(4-[2'-(2-Chloro-5-trifluoromethyl-phenoxymethyl)-b...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Prostaglandin E2 synthase-1 in IL-1beta stimulated microsomal fraction of human A549 cell assessed as PGE2 level by RP-HPLCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50339582(4-[2'-(2-Chloro-5-trifluoromethyl-phenoxymethyl)-b...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50339582(4-[2'-(2-Chloro-5-trifluoromethyl-phenoxymethyl)-b...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant 5-lipooxygenase expressed in Escherichia coli MV1190 by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed