Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL

LigandBDBM50059213(CHEMBL3393310)Copy SMILESCopy InChI

Affinity DataKi:  85nMAssay Description:Inhibition of DLK (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

Curated by ChEMBL

LigandBDBM50059213(CHEMBL3393310)Copy SMILESCopy InChI

Affinity DataIC50:  767nMAssay Description:Inhibition of human DLK transfected in HEK293 cells assessed as JNK phosphorylation after 5.5 hrs by Hoechst-33342 staining-based assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI