Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetApelin receptor(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50393896(CHEMBL2158275)
Affinity DataIC50:  3.11E+3nMAssay Description:Antagonist activity at APJ receptor expressed in CHOK1 cells assessed as inhibition of apelin13-induced beta-arrestin recruitment after 90 mins by lu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50393896(CHEMBL2158275)
Affinity DataIC50: >7.90E+4nMAssay Description:Inhibition of AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed