Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50155450(CHEMBL3779953)
Affinity DataIC50: <250nMAssay Description:Inhibition of human KDM4C preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50155450(CHEMBL3779953)
Affinity DataIC50: <250nMAssay Description:Inhibition of human PHF8 preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50155450(CHEMBL3779953)
Affinity DataIC50: <250nMAssay Description:Inhibition of human KDM5B preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 6A(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50155450(CHEMBL3779953)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human KDM6A preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2B(Homo sapiens (Human))
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50155450(CHEMBL3779953)
Affinity DataIC50: >2.50E+3nMAssay Description:Inhibition of human KDM2B preincubated for 10 mins followed by substrate addition by AlphaLISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed