Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 24 hits in this display
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
IC50: 8.51E+3nMAssay Description:Inhibition of HIF1 activation in human Hep3B cells assessed as inhibition of hypoxia-induced luciferase expression after 16 hrs by reporter assayMore data for this Ligand-Target Pair
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
IC50: 1.15E+4nMAssay Description:Inhibition of SARS-CoV PLpro expressed in Escherichia coli BL21 (DE3) using Arg-Leu-Arg-Gly-Gly-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
IC50: 1.25E+4nMAssay Description:Inhibition of HIF1 activation in human AGS cells assessed as inhibition of hypoxia-induced luciferase expression after 16 hrs by reporter assayMore data for this Ligand-Target Pair
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
IC50: 3.87E+4nMAssay Description:Inhibition of SARS-CoV 3CLpro expressed in Escherichia coli BL21 (DE3) using Dabcyl-KNSTLQSGLRKE-Edan as substrate after 60 mins by FRET analysisMore data for this Ligand-Target Pair
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)
BDBM51317(1,6-dimethylnaphtho[1,2-g][1]benzofuran-10,11-dion...)