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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
TGF-beta receptor type-1
(Homo sapiens (Human))
Abbott Laboratories
Curated by
ChEMBL
Ligand
BDBM50255959
(4-(5-fluoro-6-methylpyridin-2-yl)-5-(quinoxalin-6-...)
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Affinity Data
Ki: 0.700nM
Assay Description:
Binding affinity to human TGFBR1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
TGF-beta receptor type-1
(Homo sapiens (Human))
Abbott Laboratories
Curated by
ChEMBL
Ligand
BDBM50255959
(4-(5-fluoro-6-methylpyridin-2-yl)-5-(quinoxalin-6-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 33.5nM
Assay Description:
Inhibition of TGFBR1 (unknown origin) transfected in human HepG2 cells after 24 hrs by plasminogen activator inhibitor-luciferase reporter gene assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
TGF-beta receptor type-1
(Homo sapiens (Human))
Abbott Laboratories
Curated by
ChEMBL
Ligand
BDBM50255959
(4-(5-fluoro-6-methylpyridin-2-yl)-5-(quinoxalin-6-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.25E+4nM
Assay Description:
Inhibition of p38alpha (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI