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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetB1 bradykinin receptor(Homo sapiens (Human))
Elan Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50222683(CHEMBL398008 | N-(4-bromo-3-(2-methylthiazol-4-yl)...)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at human bradykinin B1 receptor in IL1beta stimulated IMR90 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed