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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
L-lactate dehydrogenase A chain
(Rattus norvegicus (Rat))
Astrazeneca
Ligand
BDBM86134
(LDHA Inhibitor, 30)
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Affinity Data
IC50: 2.95E+4nM
pH: 7.5 T: 2°C
Assay Description:
Enzyme assay using lactate dehydrogenase A (LDHA).
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
L-lactate dehydrogenase A chain
(Rattus norvegicus (Rat))
Astrazeneca
Ligand
BDBM86134
(LDHA Inhibitor, 30)
Copy SMILES
Copy InChI
Affinity Data
Kd: 1.20E+3nM
pH: 7.4
Assay Description:
A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI