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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86134(LDHA Inhibitor, 30)
Affinity DataIC50:  2.95E+4nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Rattus norvegicus (Rat))
Astrazeneca

LigandPNGBDBM86134(LDHA Inhibitor, 30)
Affinity DataKd:  1.20E+3nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed