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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Alpha-2A adrenergic receptor
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
ChEMBL
Ligand
BDBM50403744
(LUSAPERIDONE)
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Affinity Data
IC50: 0.550nM
Assay Description:
Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
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PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Alpha-2C adrenergic receptor
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
ChEMBL
Ligand
BDBM50403744
(LUSAPERIDONE)
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Copy InChI
Affinity Data
IC50: 1.70nM
Assay Description:
Binding affinity at human Alpha-2C adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Alpha-2B adrenergic receptor
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
ChEMBL
Ligand
BDBM50403744
(LUSAPERIDONE)
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Copy InChI
Affinity Data
IC50: 2.60nM
Assay Description:
Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
Janssen Research Foundation
Curated by
ChEMBL
Ligand
BDBM50403744
(LUSAPERIDONE)
Copy SMILES
Copy InChI
Affinity Data
IC50: 347nM
Assay Description:
Binding affinity at human Alpha-1A adrenergic receptor in CHO cells uby [3H]prazosin (0.25 nM) displacement.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI