Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
D(3) dopamine receptor
(Homo sapiens (Human))
Aptuit
Curated by
ChEMBL
Ligand
BDBM50154894
(CHEMBL3775338 | US10273244, Example 28 | US1058413...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.398nM
Assay Description:
Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation counter metho...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
D(3) dopamine receptor
(Homo sapiens (Human))
Aptuit
Curated by
ChEMBL
Ligand
BDBM50154894
(CHEMBL3775338 | US10273244, Example 28 | US1058413...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.417nM
Assay Description:
3H]-Spiperone Binding Assay at hD3 and hD4 recombinant receptors CHO cells transiently transfected with human dopamine type 3 or 4 receptors (CHO-hD3...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
D(3) dopamine receptor
(Homo sapiens (Human))
Aptuit
Curated by
ChEMBL
Ligand
BDBM50154894
(CHEMBL3775338 | US10273244, Example 28 | US1058413...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 0.417nM
Assay Description:
[3H]-Spiperone Binding Assay at hD3 and hD4 recombinant receptors CHO cells transiently transfected with human dopamine type 3 or 4 receptors (CHO-hD...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
D(2) dopamine receptor
(Homo sapiens (Human))
Aptuit
Curated by
ChEMBL
Ligand
BDBM50154894
(CHEMBL3775338 | US10273244, Example 28 | US1058413...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 10nM
Assay Description:
Displacement of [3H]-spiperone from human dopamine D2 receptor expressed in CHO-K1 cell membranes after 120 mins by liquid scintillation counter meth...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
D(2) dopamine receptor
(Homo sapiens (Human))
Aptuit
Curated by
ChEMBL
Ligand
BDBM50154894
(CHEMBL3775338 | US10273244, Example 28 | US1058413...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 10.5nM
Assay Description:
CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
D(2) dopamine receptor
(Homo sapiens (Human))
Aptuit
Curated by
ChEMBL
Ligand
BDBM50154894
(CHEMBL3775338 | US10273244, Example 28 | US1058413...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 10.5nM
Assay Description:
Functional Calcium Assay at hD2 recombinant receptor. CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to G...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
Aptuit
Curated by
ChEMBL
Ligand
BDBM50154894
(CHEMBL3775338 | US10273244, Example 28 | US1058413...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >100nM
Assay Description:
Inhibition of human ERG tail current expressed in HEK293 cells after 5 mins by patch clamp assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
UniProtKB/TrEMBL
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI