Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM50192249(CHEMBL3923578 | US10239870, Example 239)
BDBM50192249(CHEMBL3923578 | US10239870, Example 239)
Ki: 3.60nMAssay Description:Displacement of [3H]-spiperone from human dopamine D3 receptor expressed in CHO-K1 cell membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
BDBM50192249(CHEMBL3923578 | US10239870, Example 239)
Ki: 3.63nMAssay Description:[125I]-7OH-PIPAT Binding Assay at rat native D3 receptor on membranes from rat ventral striatum. Homogenates from frozen rat brain ventral striatum (...More data for this Ligand-Target Pair
BDBM50192249(CHEMBL3923578 | US10239870, Example 239)
BDBM50192249(CHEMBL3923578 | US10239870, Example 239)
BDBM50192249(CHEMBL3923578 | US10239870, Example 239)
Ki: 1.62E+3nMAssay Description:CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...More data for this Ligand-Target Pair
BDBM50192249(CHEMBL3923578 | US10239870, Example 239)
BDBM50192249(CHEMBL3923578 | US10239870, Example 239)