Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 63 hits in this display
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: <100nMAssay Description:LSD1: A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: <100nMAssay Description:LSD1: A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: <100nMpH: 8.0 T: 2°CAssay Description:A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and the m...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: <100nMpH: 8.0 T: 2°CAssay Description:A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and the m...More data for this Ligand-Target Pair
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: <100nMpH: 8.0 T: 2°CAssay Description:A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and the m...More data for this Ligand-Target Pair
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: <100nMpH: 8.0 T: 2°CAssay Description:A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and the m...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: <100nMAssay Description:A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and the m...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: 270nMAssay Description:A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and the m...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: 270nMpH: 8.0 T: 2°CAssay Description:A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and the m...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: 270nMpH: 8.0 T: 2°CAssay Description:A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and the m...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: 270nMAssay Description:LSD1: A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: 270nMpH: 8.0 T: 2°CAssay Description:A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and the m...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: 270nMpH: 8.0 T: 2°CAssay Description:A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and the m...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: 270nMAssay Description:LSD1: A test compound dissolved in DMSO was added by to a reaction solution (50 mM Tris-HCl (pH 8.0), 0.1% BSA, 1 mM DTT) containing LSD1 enzyme, and...More data for this Ligand-Target Pair
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-B inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMAssay Description:A test compound dissolved in DMSO was added to a reaction solution (100 mM HEPES (pH 7.5), 5% glycerol) containing MAO-A enzyme (Sigma-Aldrich Co. LL...More data for this Ligand-Target Pair
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMAssay Description:A test compound dissolved in DMSO was added to a reaction solution (100 mM HEPES (pH 7.5), 5% glycerol, 10% DMSO) containing MAO-B enzyme (Sigma-Aldr...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: >1.00E+5nMAssay Description:A test compound dissolved in DMSO was added to a reaction solution (100 mM HEPES (pH 7.5), 5% glycerol) containing MAO-A enzyme (Sigma-Aldrich Co. LL...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: >1.00E+5nMAssay Description:A test compound dissolved in DMSO was added to a reaction solution (100 mM HEPES (pH 7.5), 5% glycerol, 10% DMSO) containing MAO-B enzyme (Sigma-Aldr...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMAssay Description:MAO-A: The MAO-A inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test co...More data for this Ligand-Target Pair
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMAssay Description:MAO-B: The MAO-B inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test co...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: >1.00E+5nMAssay Description:MAO-A: The MAO-A inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test co...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: >1.00E+5nMAssay Description:MAO-B: The MAO-B inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test co...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMAssay Description:The MAO-A inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMAssay Description:The MAO-B inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: >1.00E+5nMAssay Description:The MAO-A inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
IC50: >1.00E+5nMAssay Description:The MAO-B inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-B inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-A inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-B inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-A inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-B inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-A inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:A test compound dissolved in DMSO was added to a reaction solution (100 mM HEPES (pH 7.5), 5% glycerol, 10% DMSO) containing MAO-B enzyme (Sigma-Aldr...More data for this Ligand-Target Pair
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:A test compound dissolved in DMSO was added to a reaction solution (100 mM HEPES (pH 7.5), 5% glycerol) containing MAO-A enzyme (Sigma-Aldrich Co. LL...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:A test compound dissolved in DMSO was added to a reaction solution (100 mM HEPES (pH 7.5), 5% glycerol, 10% DMSO) containing MAO-B enzyme (Sigma-Aldr...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:A test compound dissolved in DMSO was added to a reaction solution (100 mM HEPES (pH 7.5), 5% glycerol) containing MAO-A enzyme (Sigma-Aldrich Co. LL...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-B inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK. A test compound...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-B inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK. A test compound...More data for this Ligand-Target Pair
BDBM256699(US10053456, 79 | US10414761, Example 79 | US109682...)
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-A inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256680(US10053456, 59 | US10414761, Example 59 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-A inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
BDBM256698(US10053456, 78 | US10414761, Example 78 | US109682...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MAO-A inhibitory activity evaluation described below followed the protocol of MAO-Glo (registered trademark) Assay of Promega KK.A test compound ...More data for this Ligand-Target Pair
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