Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetType-1 angiotensin II receptor(Bos taurus)
China Pharmaceutical University

Curated by ChEMBL

LigandBDBM50387806(CHEMBL2058366)Copy SMILESCopy InChI

Affinity DataIC50:  92nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetEndothelin-1 receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

LigandBDBM50387806(CHEMBL2058366)Copy SMILESCopy InChI

Affinity DataIC50:  99nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI