Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 1 hits in this display
BDBM50345571(3-(2-(pyridin-2-yl)ethynyl)-5-chlorobenzonitrile |...)
IC50: 1.03nMAssay Description:Antagonist activity at rat mGluR5 expressed in human HEK-293 cells assessed as inhibition of glutamate-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair