Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
Johns Hopkins Medical Institutions

Curated by ChEMBL
LigandPNGBDBM50018560((+/-)-1'-(4-chlorobenzyl)-3-phenyl-3,4'-bipiperidi...)
Affinity DataIC50:  27nMAssay Description:Displacement of [3H]N-methylscopolamine from rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Johnson & Johnson Prd

Curated by ChEMBL
LigandPNGBDBM50018560((+/-)-1'-(4-chlorobenzyl)-3-phenyl-3,4'-bipiperidi...)
Affinity DataIC50:  830nMAssay Description:Antagonist activity at human CXCR3 expressed in CHO cells assessed as inhibition of ITAC-stimulated [35S]GTPgammaS binding pretreated 30 mins before ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed