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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Muscarinic acetylcholine receptor M1/M2/M3/M4/M5
(RAT)
Johns Hopkins Medical Institutions
Curated by
ChEMBL
Ligand
BDBM50018560
((+/-)-1'-(4-chlorobenzyl)-3-phenyl-3,4'-bipiperidi...)
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Affinity Data
IC50: 27nM
Assay Description:
Displacement of [3H]N-methylscopolamine from rat brain homogenate
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
C-X-C chemokine receptor type 3
(Homo sapiens (Human))
Johnson & Johnson Prd
Curated by
ChEMBL
Ligand
BDBM50018560
((+/-)-1'-(4-chlorobenzyl)-3-phenyl-3,4'-bipiperidi...)
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Copy InChI
Affinity Data
IC50: 830nM
Assay Description:
Antagonist activity at human CXCR3 expressed in CHO cells assessed as inhibition of ITAC-stimulated [35S]GTPgammaS binding pretreated 30 mins before ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI