Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM50087020(8-(5,8-Dichloro-1,2,3,4-tetrahydro-naphthalen-2-yl...)
Ki: 2.80nMAssay Description:Effective concentration required to stimulate binding of GTPgammaS to Opioid receptor like 1 was determined using scintillation proximity assayMore data for this Ligand-Target Pair
BDBM50087020(8-(5,8-Dichloro-1,2,3,4-tetrahydro-naphthalen-2-yl...)
Ki: 5.90nMAssay Description:Competitive binding displacement analyses was performed from permanently transfected HEK293 cells expressing human Opioid receptor mu 1More data for this Ligand-Target Pair
BDBM50087020(8-(5,8-Dichloro-1,2,3,4-tetrahydro-naphthalen-2-yl...)
Ki: 40nMAssay Description:Competitive binding displacement analyses was performed from permanently transfected HEK293 cells expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
BDBM50087020(8-(5,8-Dichloro-1,2,3,4-tetrahydro-naphthalen-2-yl...)
Ki: 415nMAssay Description:Competitive binding displacement analyses was performed from permanently transfected HEK293 cells expressing human Opioid receptor delta 1More data for this Ligand-Target Pair