Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50171586(CHEMBL196620 | Pyridine-2-carboxylic acid [2-(1-be...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity towards melanin-concentrating hormone receptor 1 in IMR32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50171586(CHEMBL196620 | Pyridine-2-carboxylic acid [2-(1-be...)
Affinity DataIC50:  370nMAssay Description:Inhibitory concentration against MCH1R IMR32 cells in FLIPR-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed