Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 11 hits in this display
BDBM50060725(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
BDBM50060725(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
Ki: 0.75nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
BDBM50075808(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
BDBM50060726(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
BDBM50060725(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
Ki: 1.80nMAssay Description:Ability of the compound to reverse Neuropeptide Y receptor type 1-induced inhibition of forskolin-induced inhibition of forskolin-stimulated cAMPMore data for this Ligand-Target Pair
BDBM50060726(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
BDBM50060725(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
BDBM50060726(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
BDBM50060726(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
BDBM50060725(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
BDBM50060725(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)