Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetLethal factor(Bacillus anthracis)
Burnham Institute

LigandBDBM8460(5-{[5-(4-chlorophenyl)furan-2-yl]methylidene}-2-su...)Copy SMILESCopy InChI

Affinity DataIC50:  4.40E+3nMpH: 7.4 T: 2°CAssay Description:Fluorescence peptide cleavage assay was performed in a 96-well plate. Each reaction contained MAPKKide, LF, and the small-molecule inhibitor. The C-t...More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoPurchasePC cidPC sidPatentsSimilars

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TargetProtein arginine N-methyltransferase 5(Homo sapiens (Human))
Sichuan University

LigandBDBM8460(5-{[5-(4-chlorophenyl)furan-2-yl]methylidene}-2-su...)Copy SMILESCopy InChI

Affinity DataIC50:  6.70E+4nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPurchasePC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI