Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Glucagon receptor
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50104372
(4-[2-(4-Chloro-phenyl)-5-(4-phenoxy-phenyl)-3H-imi...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 27nM
Assay Description:
Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glucagon receptor
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50104372
(4-[2-(4-Chloro-phenyl)-5-(4-phenoxy-phenyl)-3H-imi...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 110nM
Assay Description:
Affinity for human glucagon receptor in presence of Mg2+
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mitogen-activated protein kinase 11/12/13/14
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50104372
(4-[2-(4-Chloro-phenyl)-5-(4-phenoxy-phenyl)-3H-imi...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 250nM
Assay Description:
Binding affinity towards human Mitogen-activated protein kinase p38 expressed as IC50
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Glucagon receptor
(Homo sapiens (Human))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50104372
(4-[2-(4-Chloro-phenyl)-5-(4-phenoxy-phenyl)-3H-imi...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 250nM
Assay Description:
Inhibition of human glucagon receptor expressed in CHO cell membranes by radioligand displacement assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
Copy BDB DOI