Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50067113(3,4-Dichloro-N-(3-pyridin-2-yl-isoquinolin-1-yl)-b...)
Affinity DataKi:  2.10E+5nMAssay Description:Tested for antagonist activity by displacement of specific [125I]-AB-MECA binding at human Adenosine A3 receptor expressed in HEK 293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed