Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50008874(9-Chloro-2-furan-2-yl-6H-[1,2,4]triazolo[1,5-c]qui...)
Affinity DataKi:  260nMAssay Description:In vitro binding affinity at human Adenosine A3 receptor from HEK-293 cells by [125I]-AB-MECA displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50008874(9-Chloro-2-furan-2-yl-6H-[1,2,4]triazolo[1,5-c]qui...)
Affinity DataKi:  3.95E+3nMAssay Description:Displacement of [3H]-¿-PIA from Adenosine A1 receptor of rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50008874(9-Chloro-2-furan-2-yl-6H-[1,2,4]triazolo[1,5-c]qui...)
Affinity DataKi:  4.38E+3nMAssay Description:Displacement of [3H]-CGH 21680 from Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50008874(9-Chloro-2-furan-2-yl-6H-[1,2,4]triazolo[1,5-c]qui...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of binding towards adenosine A1 receptor using [3H]-N-cyclohexyladenosine ([3H]-CHA) in rat whole brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50008874(9-Chloro-2-furan-2-yl-6H-[1,2,4]triazolo[1,5-c]qui...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of binding to Adenosine-2 receptor using [3H]NECA in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed