Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 22 hits in this display
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
Ki: 5.90nMAssay Description:Binding affinity towards rat Dopamine receptor D3 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
Ki: 198nMAssay Description:Displacement of [125I]ABN from human dopamine D2L receptor expressed in HEK293 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
Ki: 198nMAssay Description:Binding affinity towards rat Dopamine receptor D2 in Sf9 cells expressing in recombinant baculovirus (Bv) using [125I]-IABN as radioligandMore data for this Ligand-Target Pair
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
IC50: 173nMAssay Description:Mitogenic stimulation or antagonism of 30 nM quinpirole-stimulated mitogenesis in CHO cells expressing human dopamine D3 receptorMore data for this Ligand-Target Pair
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)
BDBM50129429(9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichl...)