Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetArylamine N-acetyltransferase 2(Mus musculus)
University Of Oxford

Curated by ChEMBL

LigandBDBM50014926(CHEMBL3262057)Copy SMILESCopy InChI

Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair

Target InfoReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetArylamine N-acetyltransferase 1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL

LigandBDBM50014926(CHEMBL3262057)Copy SMILESCopy InChI

Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of human NAT1 assessed as rate of free thiol coenzyme A production using arylamine and AcCoA as substrate by Ellman's methodMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatentsSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI