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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMuscarinic acetylcholine receptor M1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50033160(3-(3-Chloro-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octa...)
Affinity DataIC50:  56nMAssay Description:Binding activity against muscarinic acetylcholine receptor M1 in rat brain, using [3H]OXO-M as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50033160(3-(3-Chloro-pyrazin-2-yl)-1-aza-bicyclo[2.2.2]octa...)
Affinity DataIC50:  180nMAssay Description:Binding activity against muscarinic acetylcholine receptor M1 in rat brain, using [3H]-Pz as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed