Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Oxysterols receptor LXR-beta
(Homo sapiens (Human))
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM50294738
(CHEMBL551981 | {3-[3-Benzyl-8-(trifluoromethyl)qui...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.90E+4nM
Assay Description:
Displacement of [3H]T0901317 from human recombinant N-terminal biotinylated tagged LXRbeta ligand binding domain (154-461) expressed in Escherichia c...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Oxysterols receptor LXR-alpha
(Homo sapiens (Human))
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM50294738
(CHEMBL551981 | {3-[3-Benzyl-8-(trifluoromethyl)qui...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.12E+6nM
Assay Description:
Displacement of [3H]T0901317 from human recombinant N-terminal biotinylated tagged LXRalpha ligand binding domain (197-447) expressed in Escherichia ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Oxysterols receptor LXR-beta
(Homo sapiens (Human))
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM50294738
(CHEMBL551981 | {3-[3-Benzyl-8-(trifluoromethyl)qui...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.02E+4nM
Assay Description:
Agonist activity at human LXRbeta ligand binding domain (219-462) expressed in human HuH7 cells cotransfected with Gal4-DBD by luciferase transactiva...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Oxysterols receptor LXR-alpha
(Homo sapiens (Human))
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM50294738
(CHEMBL551981 | {3-[3-Benzyl-8-(trifluoromethyl)qui...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.35E+4nM
Assay Description:
Agonist activity at human LXRalpha ligand binding domain (205-448) expressed in human HuH7 cells cotransfected with Gal4-DBD by luciferase transactiv...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI