Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 15 hits in this display
BDBM382294(US10273244, Example 171 | US10584135, Example 171)
BDBM382294(US10273244, Example 171 | US10584135, Example 171)
BDBM50154855(CHEMBL3775033 | US10273244, Example 168 | US105841...)
Ki: 9.12nMAssay Description:[3H]-Spiperone Binding Assay at hD3 and hD4 recombinant receptors CHO cells transiently transfected with human dopamine type 3 or 4 receptors (CHO-hD...More data for this Ligand-Target Pair
BDBM50154855(CHEMBL3775033 | US10273244, Example 168 | US105841...)
Ki: 9.12nMAssay Description:3H]-Spiperone Binding Assay at hD3 and hD4 recombinant receptors CHO cells transiently transfected with human dopamine type 3 or 4 receptors (CHO-hD3...More data for this Ligand-Target Pair
BDBM50154855(CHEMBL3775033 | US10273244, Example 168 | US105841...)
BDBM382295(US10273244, Example 172 | US10584135, Example 172)
Ki: 23.4nMAssay Description:3H]-Spiperone Binding Assay at hD3 and hD4 recombinant receptors CHO cells transiently transfected with human dopamine type 3 or 4 receptors (CHO-hD3...More data for this Ligand-Target Pair
BDBM382295(US10273244, Example 172 | US10584135, Example 172)
Ki: 23.4nMAssay Description:[3H]-Spiperone Binding Assay at hD3 and hD4 recombinant receptors CHO cells transiently transfected with human dopamine type 3 or 4 receptors (CHO-hD...More data for this Ligand-Target Pair
BDBM382294(US10273244, Example 171 | US10584135, Example 171)
BDBM382294(US10273244, Example 171 | US10584135, Example 171)
BDBM50154855(CHEMBL3775033 | US10273244, Example 168 | US105841...)
Ki: 617nMAssay Description:CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...More data for this Ligand-Target Pair
BDBM50154855(CHEMBL3775033 | US10273244, Example 168 | US105841...)
Ki: 617nMAssay Description:Functional Calcium Assay at hD2 recombinant receptor. CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to G...More data for this Ligand-Target Pair
BDBM50154855(CHEMBL3775033 | US10273244, Example 168 | US105841...)
BDBM382295(US10273244, Example 172 | US10584135, Example 172)
Ki: 1.20E+3nMAssay Description:CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to Gα16 protein (CHO-Gα16-hD2L) were re-suspended ...More data for this Ligand-Target Pair
BDBM382295(US10273244, Example 172 | US10584135, Example 172)
Ki: 1.20E+3nMAssay Description:Functional Calcium Assay at hD2 recombinant receptor. CHO cells stably expressing human dopamine receptor type 2, long variant (hD2L), coupled to G...More data for this Ligand-Target Pair
BDBM50154855(CHEMBL3775033 | US10273244, Example 168 | US105841...)