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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063520(CHEMBL3398533)
Affinity DataIC50:  142nMAssay Description:Inhibition of human recombinant MAO-A assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yaroslavl State Technical University

Curated by ChEMBL
LigandPNGBDBM50063520(CHEMBL3398533)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant MAO-B assessed as kynuramine oxidation to 4-hydroxyquinoline formation by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed