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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Banyu Tsukuba Research Institute
Curated by
ChEMBL
Ligand
BDBM50196291
(6-(benzo[d][1,3]dioxol-5-yl)-5-methyl-3-phenylisox...)
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Affinity Data
IC50: 26nM
Assay Description:
Antagonist activity at rat mGluR7 expressed in CHO cells assessed as inhibition of LAP-induced intracellular calcium mobilization by FLIPR
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
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Ligand Info
CHEMBL
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Article
PubMed
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Target
Nuclear receptor subfamily 4 group A member 2
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM50196291
(6-(benzo[d][1,3]dioxol-5-yl)-5-methyl-3-phenylisox...)
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Copy InChI
Affinity Data
EC50: 0.800nM
Assay Description:
Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI