Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104331(US8575186, 177 | US8575186, 178 | US8575186, 94/16...)
Affinity DataKi:  0.280nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50364980(CHEMBL1950775)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50364980(CHEMBL1950775)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104331(US8575186, 177 | US8575186, 178 | US8575186, 94/16...)
Affinity DataKi:  0.320nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104331(US8575186, 177 | US8575186, 178 | US8575186, 94/16...)
Affinity DataKi:  0.370nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50364980(CHEMBL1950775)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed