Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50400797(CHEMBL2203622)
Affinity DataIC50:  850nMAssay Description:Antagonist activity at adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50400797(CHEMBL2203622)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50400797(CHEMBL2203622)
Affinity DataIC50:  3.20E+3nMAssay Description:Antagonist activity at CHT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed