Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 34 hits in this display
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
IC50: 4nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
IC50: 4nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
IC50: 16nMAssay Description:Inhibition of dog DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
IC50: 20nMAssay Description:Inhibition of rat DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
IC50: 25nMAssay Description:Inhibition of mouse DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
Cathepsin S(Homo sapiens (Human))Charles River Discovery Research Services
Curated by ChEMBL
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
Cathepsin D(Homo sapiens (Human))Charles River Discovery Research Services
Curated by ChEMBL
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
Cathepsin G(Homo sapiens (Human))Charles River Discovery Research Services
Curated by ChEMBL
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
Cathepsin E(Homo sapiens (Human))Charles River Discovery Research Services
Curated by ChEMBL
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
Cathepsin B(Homo sapiens (Human))Charles River Discovery Research Services
Curated by ChEMBL
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
Cathepsin K(Homo sapiens (Human))Charles River Discovery Research Services
Curated by ChEMBL
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
Cathepsin Z(Homo sapiens (Human))Charles River Discovery Research Services
Curated by ChEMBL
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)
BDBM50195235(CHEMBL3900409 | US10287258, Example 2 | US10669245...)