Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50339887(1-(1-(4-(benzofuran-2-yl)pyrimidin-2-yl)piperidin-...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human FAAH assessed as hydrolysis of anandamidoaminomethylcumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Amgen

Curated by ChEMBL
LigandPNGBDBM50339887(1-(1-(4-(benzofuran-2-yl)pyrimidin-2-yl)piperidin-...)
Affinity DataIC50:  780nMAssay Description:Inhibition of rat FAAH assessed as hydrolysis of anandamidoaminomethylcumarinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed