Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM50020852(8-(4-Amino-phenyl)-1,3-dimethyl-3,7-dihydro-purine...)
BDBM50020852(8-(4-Amino-phenyl)-1,3-dimethyl-3,7-dihydro-purine...)
Ki: 130nMAssay Description:Antagonism of cyclic [3H]AMP accumulation in guinea pig cerebral cortical slices (elicited by 15 uM 2-chloroadenosine at adenosine A2 receptor)More data for this Ligand-Target Pair
BDBM50020852(8-(4-Amino-phenyl)-1,3-dimethyl-3,7-dihydro-purine...)
BDBM50020852(8-(4-Amino-phenyl)-1,3-dimethyl-3,7-dihydro-purine...)
BDBM50020852(8-(4-Amino-phenyl)-1,3-dimethyl-3,7-dihydro-purine...)
BDBM50020852(8-(4-Amino-phenyl)-1,3-dimethyl-3,7-dihydro-purine...)
IC50: 1.80nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membrane preparations using N6-[3H]-cyclohexyladenosine as a radioligandMore data for this Ligand-Target Pair