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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
1
hit in this display
Target
3-phosphoinositide-dependent protein kinase 1 [51-359]
(Homo sapiens (Human))
Sunesis Pharmaceuticals
US Patent
Ligand
BDBM282089
(3-((5-(4-aminoquinazolin- 6-yl)thiophen-2-yl)methy...)
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Affinity Data
IC50: <100nM
Assay Description:
PDK1 (amino acids 51-359) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) were expressed as N-terminally tagged GST fusi...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
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Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
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