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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50295902(3-(1-Methyl-1H-pyrrolo[3,2-b]pyridin-3-yl)-4-(1-(3...)
Affinity DataIC50:  760nMAssay Description:Inhibition of recombinant GST-GSK3beta expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50295902(3-(1-Methyl-1H-pyrrolo[3,2-b]pyridin-3-yl)-4-(1-(3...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant IKK2 expressed in Bac-to Bac baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50295902(3-(1-Methyl-1H-pyrrolo[3,2-b]pyridin-3-yl)-4-(1-(3...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant MEK1 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50295902(3-(1-Methyl-1H-pyrrolo[3,2-b]pyridin-3-yl)-4-(1-(3...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant ERK1 expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50295902(3-(1-Methyl-1H-pyrrolo[3,2-b]pyridin-3-yl)-4-(1-(3...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant PKCE expressed in Bac-to Bac baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50295902(3-(1-Methyl-1H-pyrrolo[3,2-b]pyridin-3-yl)-4-(1-(3...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of recombinant Aurora A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed