Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50424641(CHEMBL2313498)
Affinity DataEC50:  3.30E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50424641(CHEMBL2313498)
Affinity DataEC50:  3.31E+3nMAssay Description:Positive allosteric modulator activity at human muscarinic M1 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed