Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122804(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-pyrazo...)
Affinity DataKi:  45nMAssay Description:Ability to displace [3H]5-CT (1.5 nM) from HeLa cells of human 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122804(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-pyrazo...)
Affinity DataKi:  49nMAssay Description:Ability to displace [3H]5-CT (2.0 nM) from HeLa cells of human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122804(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-pyrazo...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]ketanserin (0.5 nM) from rat cerebral cortex 5-hydroxytryptamine 2A receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122804(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-pyrazo...)
Affinity DataKi:  570nMAssay Description:Displacement of [3H]spiperone (0.5 nM) from rat corpus striatum dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122804(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-pyrazo...)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]mesulergine (0.5 nM) from rat 5-hydroxytryptamine 2C receptor expressed in SR-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed