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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Adenosine receptor A3
(Homo sapiens (Human))
National University Of Singapore
Curated by
ChEMBL
Ligand
BDBM50355164
(CHEMBL1834622)
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Affinity Data
Ki: 1.71nM
Assay Description:
Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cells after 3 hrs
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Adenosine receptor A2a
(Homo sapiens (Human))
National University Of Singapore
Curated by
ChEMBL
Ligand
BDBM50355164
(CHEMBL1834622)
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Affinity Data
Ki: 987nM
Assay Description:
Displacement of [3H]NECA from human recombinant adenosine 2A receptor expressed in CHO cells after 3 hrs
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Adenosine receptor A1
(Homo sapiens (Human))
National University Of Singapore
Curated by
ChEMBL
Ligand
BDBM50355164
(CHEMBL1834622)
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Affinity Data
Ki: 5.55E+3nM
Assay Description:
Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells after 3 hrs
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Adenosine receptor A2b
(Homo sapiens (Human))
National University Of Singapore
Curated by
ChEMBL
Ligand
BDBM50355164
(CHEMBL1834622)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Antagonist activity human recombinant adenosine 2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activit...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI