Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50355164(CHEMBL1834622)
Affinity DataKi:  1.71nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50355164(CHEMBL1834622)
Affinity DataKi:  987nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine 2A receptor expressed in CHO cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50355164(CHEMBL1834622)
Affinity DataKi:  5.55E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50355164(CHEMBL1834622)
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity human recombinant adenosine 2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed