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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
47
hits in this display
Target
Cyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3nM
Assay Description:
Inhibition of CDK2/Cyclin A
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
PubMed
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Target
Cyclin-dependent kinase/G2/mitotic-specific cyclin- 1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: 6nM
Assay Description:
Inhibition of CDK1/Cyclin B
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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Article
PubMed
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Target
Cyclin-dependent kinase 5 activator 1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 10nM
Assay Description:
Inhibition of CDK5/P25
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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Article
PubMed
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Target
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: 16nM
Assay Description:
Inhibition of CDK2/Cyclin E
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
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Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: 48nM
Assay Description:
Inhibition of GSK3-beta
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Details
Article
PubMed
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Target
Mitogen-activated protein kinase 1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 226nM
Assay Description:
Inhibition of ERK2
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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Details
Article
PubMed
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Target
Cyclin-dependent kinase 4/G1/S-specific cyclin-D1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: 350nM
Assay Description:
Inhibition of CDK4/Cyclin D1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
PubMed
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Target
Aurora kinase A
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: 670nM
Assay Description:
Inhibition of Aurora A
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
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Target
Eukaryotic translation initiation factor 2-alpha kinase 3
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of PERK
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
PubMed
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Target
Serine/threonine-protein kinase pim-1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of PIM1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
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Article
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Target
Serine/threonine-protein kinase pim-2
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of PIM2
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
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antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
PubMed
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Target
Serine/threonine-protein kinase PLK1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of PLK1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proto-oncogene tyrosine-protein kinase receptor Ret
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of RET
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
PubMed
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Target
Tyrosine-protein kinase SYK
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of SYK
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
High affinity nerve growth factor receptor
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of TRKA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of VEGFR2
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase ZAP-70
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of ZAP70
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
MAP kinase-activated protein kinase 2
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of MAPKAPK2
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Hepatocyte growth factor receptor
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of MET
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
MAP kinase-interacting serine/threonine-protein kinase 2
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of MNK2
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 26
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of MST4
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase Nek6
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of NEK6
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
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Article
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of cABL
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
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Target
Activated CDC42 kinase 1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of ACK1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of AKT1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Protein-tyrosine kinase 6
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of BRK
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Eukaryotic elongation factor 2 kinase
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of EEF2K
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of EGFR
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Focal adhesion kinase 1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of FAK
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Fibroblast growth factor receptor 1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of FGFR1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of FLT3
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Insulin-like growth factor 1 receptor
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of IGF1R
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Inhibitor of nuclear factor kappa-B kinase subunit beta
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of IKK2
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
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Target
Tyrosine-protein kinase JAK1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of JAK1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase JAK3
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of JAK3
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of cKIT
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
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CHEMBL
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PubMed
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Target
Tyrosine-protein kinase Lck
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of LCK
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
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CHEMBL
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PubMed
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Target
Tyrosine-protein kinase Lyn
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of LYN
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
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CHEMBL
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Article
PubMed
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Target
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of PDK1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
GoogleScholar
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CHEMBL
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PubMed
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Target
Serine/threonine-protein kinase PAK 4
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of PAK4
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
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CHEMBL
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PubMed
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Target
Insulin receptor
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of IR
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
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CHEMBL
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Article
PubMed
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Target
Inhibitor of nuclear factor kappa-B kinase subunit alpha
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of IKK1
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
UniProtKB/SwissProt
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CHEMBL
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Target
Vascular endothelial growth factor receptor 3
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of VEGFR3
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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CHEMBL
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Target
ALK tyrosine kinase receptor
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of ALK
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
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antibodypedia
GoogleScholar
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CHEMBL
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Article
PubMed
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Target
Mitotic checkpoint serine/threonine-protein kinase BUB1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of BUB1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
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CHEMBL
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Target
Aurora kinase B
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of Aurora B
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
PubMed
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Target
Serine/threonine-protein kinase Chk1
(Homo sapiens (Human))
Nerviano Medical Sciences
Curated by
ChEMBL
Ligand
BDBM50307506
(1-Methyl-8-{[1-(phenylcarbonyl)piperidin-4-yl]amin...)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of CHK1
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI