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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50327644(1-((6-phenylpyridin-3-yl)methyl)-5-(trifluorometho...)
Affinity DataEC50:  3.80E+3nMAssay Description:Positive allosteric modulation of muscarinic M5 receptor expressed in CHO cells assessed as effect on acetylcholine-induced intracellular calcium mob...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed