Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007157((-)-1-(1-Piperidin-1-ylmethyl-3,4-dihydro-1H-isoqu...)
Affinity DataKi:  0.620nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007157((-)-1-(1-Piperidin-1-ylmethyl-3,4-dihydro-1H-isoqu...)
Affinity DataKi:  231nMAssay Description:Affinity for opioid receptor mu sitesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Zambeletti Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50007157((-)-1-(1-Piperidin-1-ylmethyl-3,4-dihydro-1H-isoqu...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity of the compound was measured on opioid receptor delta sites.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed