Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193702(CHEMBL217078 | N-(2-(2-azabicyclo[2.2.1]heptan-2-y...)
Affinity DataIC50:  1nMAssay Description:Displacement of 125I-[Phe13,Tyr19]-MCH from human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193702(CHEMBL217078 | N-(2-(2-azabicyclo[2.2.1]heptan-2-y...)
Affinity DataEC50:  150nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed