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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM241143
(US9409895, 53 | US9630945, 53)
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Affinity Data
IC50: 39nM
Assay Description:
Inhibition of ATX (unknown origin) assessed as decrease in choline release
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2
(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by
ChEMBL
Ligand
BDBM241143
(US9409895, 53 | US9630945, 53)
Copy SMILES
Copy InChI
Affinity Data
IC50: 40nM
Assay Description:
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Ataxin-2
(Homo sapiens (Human))
Novartis
US Patent
Ligand
BDBM241143
(US9409895, 53 | US9630945, 53)
Copy SMILES
Copy InChI
Affinity Data
IC50: 40nM
Assay Description:
ATX activity was determined by measurement of released choline in reactions containing ATX (10 nM), choline oxidase (0.1 U/ml), HRP (100 U/ml), ample...
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI