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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
25
hits in this display
Target
Platelet-derived growth factor receptor beta
(Mus musculus (mouse))
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 2nM
Assay Description:
Inhibition of Tel-fused PDGFRbeta in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
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Article
PubMed
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Target
High affinity nerve growth factor receptor
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 7nM
Assay Description:
Inhibition of TRKA by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
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Target
Mast/stem cell growth factor receptor Kit
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 21nM
Assay Description:
Inhibition of Tel-fused KIT in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
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PC sid
Similars
In Depth
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Article
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Target
NT-3 growth factor receptor
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 29nM
Assay Description:
Inhibition of TRKC by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Macrophage colony-stimulating factor 1 receptor
(Mus musculus (Mouse))
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 310nM
Assay Description:
Inhibition of Tel-fused FMS in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
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In Depth
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Article
PubMed
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Target
Proto-oncogene tyrosine-protein kinase receptor Ret
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 1.10E+3nM
Assay Description:
Inhibition of Tel-fused RET in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Vascular endothelial growth factor receptor 1
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 2.20E+3nM
Assay Description:
Inhibition of Tel-fused FLT1 in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
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Target
Ephrin type-B receptor 2
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 2.40E+3nM
Assay Description:
Inhibition of Tel-fused EPHB2 in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
Details
Article
PubMed
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Target
Mitogen-activated protein kinase 9
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 3.10E+3nM
Assay Description:
Inhibition of Tel-fused JNK2 in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
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PC sid
Similars
In Depth
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Article
PubMed
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Target
Tyrosine-protein kinase ZAP-70
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 4.80E+3nM
Assay Description:
Inhibition of Tel-fused ZAP70 in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Ephrin type-A receptor 3
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 5.20E+3nM
Assay Description:
Inhibition of Tel-fused EPHA3 in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Fibroblast growth factor receptor 4
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 5.40E+3nM
Assay Description:
Inhibition of Tel-fused FGFR4 in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Proto-oncogene tyrosine-protein kinase ROS
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 5.50E+3nM
Assay Description:
Inhibition of Tel-fused ROS in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Proto-oncogene tyrosine-protein kinase Src
(Mus musculus (Mouse))
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 5.50E+3nM
Assay Description:
Inhibition of Tel-fused SRC in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
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PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Insulin-like growth factor 1 receptor
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 5.60E+3nM
Assay Description:
Inhibition of Tel-fused IGF1R in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
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PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Insulin receptor
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 5.80E+3nM
Assay Description:
Inhibition of Tel-fused INSR in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
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PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Macrophage-stimulating protein receptor
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 5.80E+3nM
Assay Description:
Inhibition of Tel-fused RON in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
ALK tyrosine kinase receptor
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 5.90E+3nM
Assay Description:
Inhibition of Tel-fused ALK in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Fibroblast growth factor receptor 3
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 6.30E+3nM
Assay Description:
Inhibition of Tel-fused FGFR3 in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Tyrosine-protein kinase Lyn
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 7.10E+3nM
Assay Description:
Inhibition of Tel-fused LYN in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Cytoplasmic tyrosine-protein kinase BMX
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 7.20E+3nM
Assay Description:
Inhibition of Tel-fused BMX in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase receptor Tie-1
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 7.90E+3nM
Assay Description:
Inhibition of Tel-fused TIE1 in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Receptor-type tyrosine-protein kinase FLT3
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: 9.40E+3nM
Assay Description:
Inhibition of Tel-fused FLT3 in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Hepatocyte growth factor receptor
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Copy InChI
Affinity Data
IC50: 9.60E+3nM
Assay Description:
Inhibition of Tel-fused MET in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
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PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Tyrosine-protein kinase Fgr
(Mus musculus)
TBA
Curated by
ChEMBL
Ligand
BDBM50384726
(CHEMBL2037208)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of Tel-fused FGR in mouse BA/F3 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI