Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL

LigandBDBM50143672(8-{2-[4-(2-Trifluoromethyl-phenyl)-piperazin-1-yl]...)Copy SMILESCopy InChI

Affinity DataKi:  5.25nMAssay Description:Binding affinity to the adrenergic receptor alpha-1D of rat aortaMore data for this Ligand-Target Pair

Target InfoReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Recordati

Curated by ChEMBL

LigandBDBM50143672(8-{2-[4-(2-Trifluoromethyl-phenyl)-piperazin-1-yl]...)Copy SMILESCopy InChI

Affinity DataKi:  26.3nMAssay Description:Binding affinity to human 5-hydroxytryptamine 1A receptor was measured using [3H]-8-hydroxy-2-(di-n-propylamine) tetraline [3H]-8-OH-DPAT) as radioli...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI