Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
BDBM50004584((8-Chloro-1-trifluoromethyl-[1,2,4]triazolo[4,3-a]...)
BDBM50004584((8-Chloro-1-trifluoromethyl-[1,2,4]triazolo[4,3-a]...)
BDBM50004584((8-Chloro-1-trifluoromethyl-[1,2,4]triazolo[4,3-a]...)
Ki: 36nMAssay Description:Binding affinity against adenosine A1 receptor in guinea pig forebrain membranes using N6-[3H]cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
BDBM50004584((8-Chloro-1-trifluoromethyl-[1,2,4]triazolo[4,3-a]...)
BDBM50004584((8-Chloro-1-trifluoromethyl-[1,2,4]triazolo[4,3-a]...)
Ki: 2.10E+3nMAssay Description:Binding affinity towards adenosine A2 receptor in rat striatal membranes using N-[3H]-ethyladenosin-5''-uronamide as radioligandMore data for this Ligand-Target Pair
BDBM50004584((8-Chloro-1-trifluoromethyl-[1,2,4]triazolo[4,3-a]...)
IC50: 5.5nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
BDBM50004584((8-Chloro-1-trifluoromethyl-[1,2,4]triazolo[4,3-a]...)
IC50: 2.10E+3nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair